Chemical name: 1-((3-(6,7-dihydro-1-methyl-7-oxo-3-propyl-1H-pyrazolo(4,3-d)pyrimidin-5-yl)-4-ethoxyphenyl)sulfonyl)-4-methylpiperazine citrate
Formula: C28H38N6O11S
Anabolic activity index: not a steroid
Androgenic activity index: not a steroid
ERIACTA-100
Introduction
ERIACTA-100 is a pharmaceutical product manufactured by Ranbaxy Laboratories Ltd., containing Sildenafil Citrate as the active ingredient. Sildenafil Citrate is a potent inhibitor of phosphodiesterase type 5 (PDE5), primarily used to treat erectile dysfunction (ED) in men. This detailed product description explores the formulation, mechanism of action, dosage, benefits, and safety considerations associated with ERIACTA-100.
Composition and Formulation
Each tablet of ERIACTA-100 contains 100mg of Sildenafil Citrate, the active ingredient responsible for its therapeutic effects. Sildenafil Citrate works by enhancing the effects of nitric oxide (NO), a chemical that relaxes smooth muscles in the penis during sexual stimulation. This relaxation allows increased blood flow into the penis, resulting in an erection sufficient for sexual activity.
The tablets are formulated using pharmaceutical-grade ingredients to ensure potency, stability, and efficacy. Inactive ingredients may include microcrystalline cellulose, calcium hydrogen phosphate (anhydrous), croscarmellose sodium, magnesium stearate, hypromellose, titanium dioxide (E171), lactose monohydrate, triacetin, and indigo carmine aluminium lake (E132) as colorant.
Mechanism of Action
Sildenafil Citrate, a selective inhibitor of PDE5, prevents the breakdown of cyclic guanosine monophosphate (cGMP) within the corpus cavernosum of the penis. During sexual stimulation, nitric oxide released from nerve endings and endothelial cells activates guanylate cyclase, leading to an increased synthesis of cGMP. Elevated levels of cGMP promote smooth muscle relaxation, allowing increased blood flow into the penile arteries and the corpora cavernosa, facilitating an erection.
Usage and Dosage
ERIACTA-100 is indicated for the treatment of erectile dysfunction in adult men. The recommended dosage is one 100mg tablet taken orally, as needed, approximately 30 to 60 minutes before anticipated sexual activity. The tablet should be swallowed whole with a full glass of water. Avoid consuming large meals or high-fat foods before taking ERIACTA-100, as these may delay the onset of action.
Dosage adjustments may be necessary based on individual response and tolerability. It is important not to exceed one tablet within a 24-hour period to avoid potential side effects and complications.
Benefits of ERIACTA-100
ERIACTA-100 offers several advantages for the treatment of ED:
- Effective Treatment: Sildenafil Citrate is a well-established treatment for erectile dysfunction, with a high success rate in improving erectile function and sexual satisfaction.
- Rapid Onset: The tablet formulation allows for rapid absorption, with onset of action typically within 30 to 60 minutes after ingestion.
- Long Duration: Effects of ERIACTA-100 may last up to 4 to 6 hours, providing a sufficient window of opportunity for sexual activity.
- Convenience: The tablet form is convenient and discreet, allowing for easy administration without the need for special preparations.
Potential Side Effects
While generally well-tolerated, ERIACTA-100 may cause side effects in some individuals. Common side effects include:
- Headache
- Flushing (reddening and warmth of the face and neck)
- Indigestion
- Nasal congestion
- Dizziness
- Blurred vision
These side effects are usually mild and transient, resolving on their own as the body adjusts to the medication. However, if these symptoms persist or worsen, medical attention may be required.
Rare but serious side effects of Sildenafil Citrate include:
- Priapism (prolonged and painful erection lasting more than 4 hours)
- Sudden decrease or loss of vision
- Sudden decrease or loss of hearing
- Chest pain or discomfort
- Allergic reactions (e.g., rash, itching, swelling of the face or throat, severe dizziness)
If any of these severe side effects occur, discontinue use of ERIACTA-100 and seek immediate medical attention.
Precautions and Warnings
Before using ERIACTA-100, it is essential to consider the following precautions:
- Medical History: Inform your healthcare provider of any existing medical conditions, especially cardiovascular diseases, kidney or liver problems, bleeding disorders, and anatomical deformities of the penis.
- Medication Interactions: Sildenafil Citrate can interact with certain medications, including nitrates (used for chest pain) and alpha-blockers (used for hypertension). These interactions can lead to severe hypotension (low blood pressure) and other complications. Therefore, avoid concurrent use with these medications unless directed by a healthcare provider.
- Alcohol and Grapefruit Juice: Limit alcohol consumption and avoid grapefruit juice while taking ERIACTA-100, as they may increase the risk of side effects or reduce the efficacy of the medication.
- Allergies: Do not use ERIACTA-100 if you are allergic to Sildenafil Citrate or any of the tablet’s ingredients.
Storage and Handling
Store ERIACTA-100 tablets in their original packaging at room temperature, away from moisture and direct sunlight. Keep out of reach of children and pets. Do not use tablets past their expiration date, and dispose of any unused medication properly.
Conclusion
ERIACTA-100 (Sildenafil Citrate Tablets) 100mg, manufactured by Ranbaxy Laboratories Ltd., is a trusted and effective medication for the treatment of erectile dysfunction. Its formulation, containing pharmaceutical-grade Sildenafil Citrate, ensures reliability and efficacy in improving erectile function and enhancing sexual performance. However, it is essential to use this medication responsibly and under the guidance of a healthcare provider to maximize benefits and minimize risks.
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